About the Authors

Lieselotte Vande Walle

Roles Conceptualization, Formal analysis, Investigation, Methodology, Writing – original draft, Writing – review & editing

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium, Discovery Sciences, Janssen Research & Development, Pharmaceutical Companies of Johnson & Johnson, Beerse, Belgium

Irma B. Stowe

Roles Data curation, Formal analysis, Investigation, Methodology, Validation, Visualization

Affiliation Department of Physiological Chemistry, Genentech, South San Francisco, California, United States of America

Pavel Šácha

Roles Data curation, Formal analysis, Investigation, Methodology, Visualization

Affiliation Institute of Organic Chemistry and Biochemistry of The Czech Academy of Sciences, Prague, Czech Republic

Bettina L. Lee

Roles Data curation, Formal analysis, Investigation, Validation, Visualization

Affiliation Department of Physiological Chemistry, Genentech, South San Francisco, California, United States of America

Dieter Demon

Roles Formal analysis, Investigation, Methodology

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium

Amelie Fossoul

Roles Formal analysis, Investigation, Methodology

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium

Filip Van Hauwermeiren

Roles Formal analysis, Investigation, Methodology

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium, Janssen Immunosciences, World Without Disease Accelerator, Pharmaceutical Companies of Johnson & Johnson, Beerse, Belgium

Pedro H. V. Saavedra

Roles Formal analysis, Investigation, Methodology

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium

Petr Šimon

Roles Formal analysis, Investigation, Methodology

Affiliation Institute of Organic Chemistry and Biochemistry of The Czech Academy of Sciences, Prague, Czech Republic

Vladimír Šubrt

Roles Conceptualization, Methodology, Resources, Validation

Affiliation Institute of Macromolecular Chemistry, Academy of Science of the Czech Republic, Prague, Czech Republic

Libor Kostka

Roles Investigation, Methodology

Affiliation Institute of Macromolecular Chemistry, Academy of Science of the Czech Republic, Prague, Czech Republic

Craig E. Stivala

Roles Investigation, Methodology, Supervision, Visualization, Writing – review & editing

Affiliation Department of Discovery Chemistry, Genentech, South San Francisco, California, United States of America

Victoria C. Pham

Roles Investigation, Methodology

Affiliation Department of Discovery Chemistry, Genentech, South San Francisco, California, United States of America

Steven T. Staben

Roles Investigation, Methodology

Affiliation Department of Discovery Chemistry, Genentech, South San Francisco, California, United States of America

Sayumi Yamazoe

Roles Investigation, Methodology

Affiliation Department of Discovery Chemistry, Genentech, South San Francisco, California, United States of America

Jan Konvalinka

Roles Conceptualization, Formal analysis, Funding acquisition, Methodology, Resources, Writing – review & editing

Affiliation Institute of Organic Chemistry and Biochemistry of The Czech Academy of Sciences, Prague, Czech Republic

Nobuhiko Kayagaki

Roles Conceptualization, Data curation, Formal analysis, Methodology, Project administration, Resources, Supervision, Visualization, Writing – review & editing

kayagaki.nobuhiko@gene.com (NK); mlamkanf@its.jnj.com (ML)

Affiliation Department of Physiological Chemistry, Genentech, South San Francisco, California, United States of America

Mohamed Lamkanfi

Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing

kayagaki.nobuhiko@gene.com (NK); mlamkanf@its.jnj.com (ML)

Affiliations Inflammation Research Center, VIB, Ghent, Belgium, Department of Internal Medicine and Pediatrics, Ghent University, Ghent, Belgium, Janssen Immunosciences, World Without Disease Accelerator, Pharmaceutical Companies of Johnson & Johnson, Beerse, Belgium

Competing Interests

LVW, FVH, and ML are employees of Janssen Pharmaceutica. IBS, BLL, CES, VCP, STS, SY, and NK are employees of Genentech. The authors declare no competing financial interests.