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Open Access
Peer-reviewed
Research Article
High Content Screening Identifies Decaprenyl-Phosphoribose 2′ Epimerase as a Target for Intracellular Antimycobacterial Inhibitors
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Thierry Christophe,
Affiliation Screening Technologies and Pharmacology, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Mary Jackson,
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Hee Kyoung Jeon,
Affiliation Screening Technologies and Pharmacology, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Denis Fenistein,
Affiliation Image Mining, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Monica Contreras-Dominguez,
Affiliation Biology of Intracellular Pathogens Inserm Avenir Group, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Jaeseung Kim,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Auguste Genovesio,
Affiliation Image Mining, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Jean-Philippe Carralot,
Affiliation Biology of Intracellular Pathogens Inserm Avenir Group, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Fanny Ewann,
Affiliation Biology of Intracellular Pathogens Inserm Avenir Group, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Eun Hye Kim,
Affiliation Biology of Intracellular Pathogens Inserm Avenir Group, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Sae Yeon Lee,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Sunhee Kang,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Min Jung Seo,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Eun Jung Park,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Henrieta Škovierová,
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Ha Pham,
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Giovanna Riccardi,
Affiliation Dipartimento di Genetica e Microbiologia, Università degli Studi di Pavia, Pavia, Italy
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Ji Youn Nam,
Affiliation Screening Technologies and Pharmacology, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Laurent Marsollier,
Affiliation Groupe d'Etude des Interactions Hôte Pathogène, Université d'Angers, Angers, France
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Marie Kempf,
Affiliation Groupe d'Etude des Interactions Hôte Pathogène, Université d'Angers, Angers, France
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Marie-Laure Joly-Guillou,
Affiliation Groupe d'Etude des Interactions Hôte Pathogène, Université d'Angers, Angers, France
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Taegwon Oh,
Affiliation International Tuberculosis Research Center, Masan, Korea
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Won Kyung Shin,
Affiliation International Tuberculosis Research Center, Masan, Korea
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Zaesung No,
Affiliation Medicinal Chemistry, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Ulf Nehrbass,
Affiliation Screening Technologies and Pharmacology, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea
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Roland Brosch,
Affiliation Institut Pasteur, Integrated Mycobacterial Pathogenomics, Paris, France
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Stewart T. Cole,
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
⨯ - [ ... ],
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Priscille Brodin
* E-mail: pbrodin@ip-korea.org
Affiliations Biology of Intracellular Pathogens Inserm Avenir Group, Institut Pasteur Korea, Bundang-gu, Seongnam-si, Gyeonggi-do, Korea, Institut Pasteur, Integrated Mycobacterial Pathogenomics, Paris, France
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High Content Screening Identifies Decaprenyl-Phosphoribose 2′ Epimerase as a Target for Intracellular Antimycobacterial Inhibitors
- Thierry Christophe,
- Mary Jackson,
- Hee Kyoung Jeon,
- Denis Fenistein,
- Monica Contreras-Dominguez,
- Jaeseung Kim,
- Auguste Genovesio,
- Jean-Philippe Carralot,
- Fanny Ewann,
- Eun Hye Kim
- Published: October 30, 2009
- https://doi.org/10.1371/journal.ppat.1000645