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Open Access
Peer-reviewed
Research Article
2-aminoimidazoles potentiate ß-lactam antimicrobial activity against Mycobacterium tuberculosis by reducing ß-lactamase secretion and increasing cell envelope permeability
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Albert B. Jeon,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Andrés Obregón-Henao,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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David F. Ackart,
Roles Conceptualization, Methodology, Resources
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Brendan K. Podell,
Roles Conceptualization, Writing – review & editing
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Juan M. Belardinelli,
Roles Data curation, Methodology, Visualization
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Mary Jackson,
Roles Conceptualization, Methodology, Supervision, Validation, Writing – review & editing
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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Tuan V. Nguyen,
Roles Data curation, Formal analysis, Investigation, Methodology, Validation
Affiliation Department of Chemistry, North Carolina State University, Raleigh, North Carolina, United States of America
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Meghan S. Blackledge,
Roles Data curation, Methodology, Resources
Affiliation Department of Chemistry, High Point University, High Point, North Carolina, United States of America
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Roberta J. Melander,
Roles Conceptualization, Investigation, Resources, Validation, Writing – review & editing
Affiliation Department of Chemistry, North Carolina State University, Raleigh, North Carolina, United States of America
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Christian Melander,
Roles Conceptualization, Data curation, Formal analysis, Project administration, Resources, Supervision, Validation, Visualization, Writing – review & editing
Affiliation Department of Chemistry, North Carolina State University, Raleigh, North Carolina, United States of America
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Benjamin K. Johnson,
Roles Data curation, Formal analysis, Validation, Visualization, Writing – review & editing
Affiliation Department of Microbiology and Molecular Genetics, Michigan State University, East Lansing, Michigan, United States of America
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Robert B. Abramovitch,
Roles Data curation, Formal analysis, Funding acquisition, Methodology, Validation, Visualization, Writing – review & editing
Affiliation Department of Microbiology and Molecular Genetics, Michigan State University, East Lansing, Michigan, United States of America
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Randall J. Basaraba
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Project administration, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
* E-mail: randall.basaraba@colostate.edu
Affiliation Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, Colorado, United States of America
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2-aminoimidazoles potentiate ß-lactam antimicrobial activity against Mycobacterium tuberculosis by reducing ß-lactamase secretion and increasing cell envelope permeability
- Albert B. Jeon,
- Andrés Obregón-Henao,
- David F. Ackart,
- Brendan K. Podell,
- Juan M. Belardinelli,
- Mary Jackson,
- Tuan V. Nguyen,
- Meghan S. Blackledge,
- Roberta J. Melander,
- Christian Melander
- Published: July 27, 2017
- https://doi.org/10.1371/journal.pone.0180925