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Open Access
Peer-reviewed
Research Article
Phenotypic, chemical and functional characterization of cyclic nucleotide phosphodiesterase 4 (PDE4) as a potential anthelmintic drug target
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Thavy Long ,
Contributed equally to this work with: Thavy Long, Liliana Rojo-Arreola
Current address: Institut National de la Recherche en Agronomie, TOXALIM UMR 1331, Toulouse, France
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Liliana Rojo-Arreola ,
Contributed equally to this work with: Thavy Long, Liliana Rojo-Arreola
Current address: CONACYT- Centro de Investigaciones Biológicas del Noroeste, La Paz, Baja California Sur, México
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Da Shi,
Affiliation Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
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Nelly El-Sakkary,
Affiliation Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
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Kurt Jarnagin,
Affiliation Anacor Pharmaceuticals, Inc., Palo Alto, California, United States of America
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Fernando Rock,
Affiliation Anacor Pharmaceuticals, Inc., Palo Alto, California, United States of America
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Maliwan Meewan,
Affiliation Anacor Pharmaceuticals, Inc., Palo Alto, California, United States of America
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Alberto A. Rascón Jr.,
Current address: Department of Chemistry, San Jose State University, San Jose, California, United States of America
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Lin Lin,
Affiliation Department of Physiology, University of California San Francisco, San Francisco, California, United States of America
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Katherine A. Cunningham,
Current address: Undergraduate Advising and Research, Stanford University, Stanford, California, United States of America
Affiliation Department of Physiology, University of California San Francisco, San Francisco, California, United States of America
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George A. Lemieux,
Affiliation Department of Physiology, University of California San Francisco, San Francisco, California, United States of America
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Larissa Podust,
Current address: Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Ruben Abagyan,
Affiliation Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
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Kaveh Ashrafi,
Affiliation Department of Physiology, University of California San Francisco, San Francisco, California, United States of America
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James H. McKerrow,
Current address: Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Conor R. Caffrey
* E-mail: ccaffrey@ucsd.edu
Current address: Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California, United States of America
Affiliations Center for Discovery and Innovation in Parasitic Diseases, University of California San Francisco, San Francisco, California, United States of America, Department of Pathology, University of California San Francisco, San Francisco, California, United States of America
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Phenotypic, chemical and functional characterization of cyclic nucleotide phosphodiesterase 4 (PDE4) as a potential anthelmintic drug target
- Thavy Long,
- Liliana Rojo-Arreola,
- Da Shi,
- Nelly El-Sakkary,
- Kurt Jarnagin,
- Fernando Rock,
- Maliwan Meewan,
- Alberto A. Rascón Jr.,
- Lin Lin,
- Katherine A. Cunningham
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- Published: July 13, 2017
- https://doi.org/10.1371/journal.pntd.0005680