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Open Access
Peer-reviewed
Research Article
Naphthoquinone Derivatives Exert Their Antitrypanosomal Activity via a Multi-Target Mechanism
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Simone Pieretti ,
Contributed equally to this work with: Simone Pieretti, Jurgen R. Haanstra
Affiliations Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy, Pharmaceutical Biochemistry Group, School of Pharmaceutical Sciences, University of Geneva, University of Lausanne, Geneva, Switzerland, Department of Biochemistry, University of Bologna, Bologna, Italy
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Jurgen R. Haanstra ,
Contributed equally to this work with: Simone Pieretti, Jurgen R. Haanstra
Affiliations Department of Pediatrics, Centre for Liver, Digestive and Metabolic Diseases, University of Groningen, University Medical Centre Groningen, Groningen, The Netherlands, Department of Molecular Cell Physiology, Faculty of Earth and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, The Netherlands
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Muriel Mazet,
Current address: Centre de Résonance Magnétique des Systèmes Biologiques (RMSB), UMR 5536 CNRS, Université Victor Segalen Bordeaux 2, Bordeaux, France
Affiliation Research Unit for Tropical Diseases, de Duve Institute and Laboratory of Biochemistry, Université Catholique de Louvain, Brussels, Belgium
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Remo Perozzo,
Affiliation Pharmaceutical Biochemistry Group, School of Pharmaceutical Sciences, University of Geneva, University of Lausanne, Geneva, Switzerland
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Christian Bergamini,
Affiliation Department of Biochemistry, University of Bologna, Bologna, Italy
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Federica Prati,
Affiliations Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy, Department of Drug Discovery and Development, Istituto Italiano di Tecnologia, Genova, Italy
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Romana Fato,
Affiliation Department of Biochemistry, University of Bologna, Bologna, Italy
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Giorgio Lenaz,
Affiliation Department of Biochemistry, University of Bologna, Bologna, Italy
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Giovanni Capranico,
Affiliation Department of Biochemistry, University of Bologna, Bologna, Italy
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Reto Brun,
Affiliation Swiss Tropical Institute, Basel, Switzerland
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Barbara M. Bakker,
Affiliations Department of Pediatrics, Centre for Liver, Digestive and Metabolic Diseases, University of Groningen, University Medical Centre Groningen, Groningen, The Netherlands, Department of Molecular Cell Physiology, Faculty of Earth and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, The Netherlands
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Paul A. M. Michels,
Affiliation Research Unit for Tropical Diseases, de Duve Institute and Laboratory of Biochemistry, Université Catholique de Louvain, Brussels, Belgium
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Leonardo Scapozza,
Affiliation Pharmaceutical Biochemistry Group, School of Pharmaceutical Sciences, University of Geneva, University of Lausanne, Geneva, Switzerland
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Maria Laura Bolognesi ,
* E-mail: marialaura.bolognesi@unibo.it (MLB); andrea.cavalli@unibo.it (AC)
Affiliation Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy
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Andrea Cavalli
* E-mail: marialaura.bolognesi@unibo.it (MLB); andrea.cavalli@unibo.it (AC)
Affiliations Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy, Department of Drug Discovery and Development, Istituto Italiano di Tecnologia, Genova, Italy
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Naphthoquinone Derivatives Exert Their Antitrypanosomal Activity via a Multi-Target Mechanism
- Simone Pieretti,
- Jurgen R. Haanstra,
- Muriel Mazet,
- Remo Perozzo,
- Christian Bergamini,
- Federica Prati,
- Romana Fato,
- Giorgio Lenaz,
- Giovanni Capranico,
- Reto Brun
- Published: January 17, 2013
- https://doi.org/10.1371/journal.pntd.0002012